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6V0X

Crystal structure of the bromodomain of human BRD9 bound to sunitinib

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue B49 A 301
ChainResidue
APHE160
AARG217
ATYR222
AHOH406
AVAL165
AILE169
ATYR173
AILE176
AASP188
AALA212
ATYR215
AASN216

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsSITE: Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding => ECO:0000269|PubMed:26365797
ChainResidueDetails
AILE169
ATYR222

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0000250|UniProtKB:Q3UQU0
ChainResidueDetails
AGLY172

224004

PDB entries from 2024-08-21

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