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6V0X

Crystal structure of the bromodomain of human BRD9 bound to sunitinib

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue B49 A 301
ChainResidue
APHE160
AARG217
ATYR222
AHOH406
AVAL165
AILE169
ATYR173
AILE176
AASP188
AALA212
ATYR215
AASN216

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsRegion: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsSite: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

244349

PDB entries from 2025-11-05

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