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6UDY

X-ray co-crystal structure of compound 5 with Mcl-1

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
B0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue Q54 A 401
ChainResidue
APHE228
AHOH534
AVAL249
AMET250
AVAL253
AARG263
ATHR266
ALEU267
APHE270
ALEU290

site_idAC2
Number of Residues10
Detailsbinding site for residue Q54 B 401
ChainResidue
BPHE228
BVAL249
BMET250
BVAL253
BARG263
BTHR266
BLEU267
BPHE270
BLEU290
BHOH532

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)
ChainResidueDetails
ALYS194
ALYS197
BLYS194
BLYS197

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PDB entries from 2025-06-11

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