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6T4I

ROR(gamma)t ligand binding domain in complex with cholesterol and allosteric ligand MRL871

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue CLR A 601
ChainResidue
AGLN286
ACYS320
AHIS323
AMET365
ALEU396
AHIS479
ALEU483
AGOL603
AHOH729

site_idAC2
Number of Residues15
Detailsbinding site for residue 4F1 A 602
ChainResidue
ALEU324
ATHR325
AILE328
AGLN329
ALEU353
ALYS354
AMET358
ALEU483
AGLN484
AGLN487
AALA496
AALA497
APHE498
ALEU505
APHE506

site_idAC3
Number of Residues5
Detailsbinding site for residue GOL A 603
ChainResidue
AHIS323
APHE377
APHE378
AGLU379
ACLR601

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsMotif: {"description":"AF-2"}
ChainResidueDetails

250835

PDB entries from 2026-03-18

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