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6SQE

Crystal structure of CREBBP bromodomain complexed with KD341

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue LSZ A 1201
ChainResidue
APRO1106
APHE1177
ASER1179
AHOH1313
AHOH1376
AHOH1386
AHOH1396
AHOH1401
AHOH1431
ALEU1109
APRO1110
AGLN1113
AVAL1115
ALEU1120
AASN1168
AARG1173
AVAL1174

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 1202
ChainResidue
AGLN1092
AASP1124
AILE1128
AHOH1331

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

220472

PDB entries from 2024-05-29

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