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6S5K

LXRbeta ligand binding domain in complex with small molecule inhibitors

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006629biological_processlipid metabolic process
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue KWE A 501
ChainResidue
APHE268
ALEU345
AHIS435
ALEU442
ALEU449
ATRP457
APHE271
ATHR272
AALA275
ASER278
AGLU315
ATHR316
APHE329
AALA343

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0000269|PubMed:20159957
ChainResidueDetails
ALYS410
ALYS448

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PDB entries from 2024-07-17

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