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6R0K

X-ray structure of Danio rerio histone deacetylase 6 (HDAC6) CD2 in complex with a inhibitor SS208

Functional Information from GO Data
ChainGOidnamespacecontents
A0000118cellular_componenthistone deacetylase complex
A0004407molecular_functionhistone deacetylase activity
A0006325biological_processchromatin organization
A0016575biological_processhistone deacetylation
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 2001
ChainResidue
AASP612
AHIS614
AASP705
AJNN2004

site_idAC2
Number of Residues5
Detailsbinding site for residue K A 2002
ChainResidue
AASP610
AASP612
AHIS614
ASER633
ALEU634

site_idAC3
Number of Residues6
Detailsbinding site for residue K A 2003
ChainResidue
APHE623
AASP626
AVAL629
ATYR662
AHOH2212
AHOH2254

site_idAC4
Number of Residues16
Detailsbinding site for residue JNN A 2004
ChainResidue
AHIS463
APRO464
ASER531
AHIS573
AHIS574
AGLY582
APHE583
AARG601
AASP612
AHIS614
APHE643
AASP705
ALEU712
ATYR745
AZN2001
AHOH2261

site_idAC5
Number of Residues7
Detailsbinding site for residue SCN A 2005
ChainResidue
AASN457
AHIS463
AARG520
ASER531
AILE532
APHE533
ASCN2007

site_idAC6
Number of Residues5
Detailsbinding site for residue SCN A 2006
ChainResidue
ATRP459
ATRP459
APRO519
AASN523
AASN523

site_idAC7
Number of Residues7
Detailsbinding site for residue SCN A 2007
ChainResidue
AARG524
AASP527
AILE532
ASCN2005
AHOH2173
AHOH2233
AHOH2331

site_idAC8
Number of Residues8
Detailsbinding site for residue SCN A 2008
ChainResidue
ASER475
AGLU478
AARG660
AHOH2115
AHOH2131
AHOH2265
AHOH2338
AHOH2444

site_idAC9
Number of Residues8
Detailsbinding site for residue SCN A 2009
ChainResidue
AGLN620
AGLU624
ALYS653
AVAL654
AGLY655
AASN663
AHOH2149
AHOH2359

site_idAD1
Number of Residues6
Detailsbinding site for residue SCN A 2010
ChainResidue
AGLN554
ATHR558
AGLN560
AASP639
AHOH2283
AHOH2358

site_idAD2
Number of Residues3
Detailsbinding site for residue SCN A 2011
ChainResidue
ASER505
ALYS506
ASER731

site_idAD3
Number of Residues3
Detailsbinding site for residue SCN A 2012
ChainResidue
AARG451
AALA491
AHOH2368

221051

PDB entries from 2024-06-12

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