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6QFQ

Structure of human Mcl-1 in complex with indole acid inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003824molecular_functioncatalytic activity
A0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue J3E A 401
ChainResidue
AHIS224
AHOH501
AHOH506
AHOH562
AALA227
APHE228
AMET250
AVAL253
AARG263
ALEU267
APHE270
AGLY271

site_idAC2
Number of Residues13
Detailsbinding site for residue J3E A 402
ChainResidue
AVAL220
AHIS224
AMET231
ASER245
AARG248
AVAL249
AHIS252
AASN260
AGLY262
AARG263
APHE318
APHE319
AHOH521

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)
ChainResidueDetails
ALYS197
ALYS194

218500

PDB entries from 2024-04-17

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