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6P6L

HCV NS3/4A protease domain of genotype 1a in complex with glecaprevir

Functional Information from GO Data
ChainGOidnamespacecontents
A0006508biological_processproteolysis
A0008236molecular_functionserine-type peptidase activity
A0019087biological_processtransformation of host cell by virus
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue EDO A 1201
ChainResidue
ALYS989
ATHR1040
AGLN1041
AARG1062
AHOH1345
AHOH1405

site_idAC2
Number of Residues3
Detailsbinding site for residue EDO A 1202
ChainResidue
AARG1109
AHOH1321
AHOH1395

site_idAC3
Number of Residues5
Detailsbinding site for residue EDO A 1203
ChainResidue
ATHR1177
ATHR1178
AMET1179
AHOH1314
AHOH1333

site_idAC4
Number of Residues1
Detailsbinding site for residue EDO A 1204
ChainResidue
AARG1011

site_idAC5
Number of Residues10
Detailsbinding site for residue SO4 A 1205
ChainResidue
ATYR1006
AGLN1008
ATYR1056
AHOH1334
AHOH1379
AHOH1400
AHOH1418
AHOH1428
AHOH1441
AHOH1475

site_idAC6
Number of Residues7
Detailsbinding site for residue SO4 A 1206
ChainResidue
ALYS1080
AARG1155
AILE1170
APRO1171
ASER1174
AHOH1301
AHOH1458

site_idAC7
Number of Residues4
Detailsbinding site for residue ZN A 1207
ChainResidue
ACYS1097
ACYS1099
ACYS1145
AHIS1149

site_idAC8
Number of Residues23
Detailsbinding site for residue O31 A 1208
ChainResidue
AHIS982
AGLN1041
ATHR1042
APHE1043
AHIS1057
AASP1081
AARG1123
AILE1132
ALEU1135
ALYS1136
AGLY1137
ASER1138
ASER1139
APHE1154
AARG1155
AALA1156
AALA1157
AHOH1376
AHOH1423
AHOH1424
AHOH1450
AHOH1451
AHOH1463

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsACT_SITE: Charge relay system; for serine protease NS3 activity => ECO:0000255|PROSITE-ProRule:PRU01166
ChainResidueDetails
AHIS1057
AASP1081
ASER1139

site_idSWS_FT_FI2
Number of Residues4
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU01166
ChainResidueDetails
ACYS1097
ACYS1099
ACYS1145
AHIS1149

224004

PDB entries from 2024-08-21

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