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6OGP

X-ray crystal structure of wild type HIV-1 protease in complex with GRL-063

Functional Information from GO Data
ChainGOidnamespacecontents
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue EDO A 101
ChainResidue
ALYS14
AGLY16
AGLY17
ALEU63

site_idAC2
Number of Residues21
Detailsbinding site for residue MJD A 102
ChainResidue
AASP29
AASP29
AASP30
AASP30
AILE47
AILE47
AGLY48
AGLY48
AGLY49
AGLY49
AILE50
APRO81
AVAL82
AVAL82
AHOH202
AHOH202
AASP25
AASP25
AGLY27
AGLY27
AALA28

Functional Information from PROSITE/UniProt
site_idPS00141
Number of Residues12
DetailsASP_PROTEASE Eukaryotic and viral aspartyl proteases active site. ALLDTGADDTVL
ChainResidueDetails
AALA22-LEU33

225946

PDB entries from 2024-10-09

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