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6NZR

CRYSTAL STRUCTURE OF TYROSINE KINASE 2 JH2 (PSEUDO KINASE DOMAIN) COMPLEXED WITH Compound_12 AKA 4-[(2-methanesulfonylphenyl)amino]-N-(H3)methyl-6-[(pyridin-2- yl)amino]pyridazine-3-carboxamide

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
B0004672molecular_functionprotein kinase activity
B0005524molecular_functionATP binding
B0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue LAJ A 901
ChainResidue
ALEU595
AARG738
AASN739
ALEU741
ASER758
AVAL640
ALYS642
ATHR687
AGLU688
ATYR689
AVAL690
AGLU691
AGLY693

site_idAC2
Number of Residues7
Detailsbinding site for residue SO4 A 902
ChainResidue
AARG744
AGLY750
ATHR751
ASER752
AHOH1007
AHOH1009
BARG744

site_idAC3
Number of Residues12
Detailsbinding site for residue LAJ B 901
ChainResidue
BLEU595
BVAL640
BLYS642
BTHR687
BGLU688
BVAL690
BGLU691
BGLY693
BARG738
BASN739
BLEU741
BSER758

site_idAC4
Number of Residues5
Detailsbinding site for residue SO4 B 902
ChainResidue
AARG744
BHIS692
BARG744
BLEU745
BGLY746

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphotyrosine => ECO:0000250|UniProtKB:Q9R117
ChainResidueDetails
ATYR604
BTYR604

222036

PDB entries from 2024-07-03

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