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6NZQ

CRYSTAL STRUCTURE OF TYROSINE KINASE 2 JH2 (PSEUDO KINASE DOMAIN) COMPLEXED WITH Compound_29 AKA 6-[(5-FLUORO-4-METH YLPYRIDIN-2-YL)AMINO]-4-({2-METHOXY-3-[(PYRIDIN-2-YLMETHYL )CARBAMOYL]PHENYL}AMINO)-N-METHYLPYRIDINE-3-CARBOXAMIDE

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
B0004672molecular_functionprotein kinase activity
B0005524molecular_functionATP binding
B0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue LB4 A 4000
ChainResidue
ALEU595
AGLU691
AGLY693
AARG738
AASN739
ALEU741
ASER758
AHOH4125
AGLY598
AVAL603
AVAL640
ALYS642
ATHR687
AGLU688
ATYR689
AVAL690

site_idAC2
Number of Residues14
Detailsbinding site for residue LB4 B 4000
ChainResidue
BLEU595
BGLY598
BVAL640
BLYS642
BTHR687
BGLU688
BTYR689
BVAL690
BGLU691
BGLY693
BARG738
BASN739
BLEU741
BSER758

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphotyrosine => ECO:0000250|UniProtKB:Q9R117
ChainResidueDetails
ATYR604
BTYR604

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PDB entries from 2024-07-17

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