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6NZP

CRYSTAL STRUCTURE OF TYROSINE KINASE 2 JH2 (PSEUDO KINASE DOMAIN) COMPLEXED WITH COMPOUND-11 AKA 6-CYCLOPROPANEAMIDO-4-{[2-METHOXY-3-(1-METHYL-1H-1,2,4-TRI AZOL-3-YL)PHENYL]AMINO}-N-(?H?)METHYLPYRIDAZINE-3-CARBOXAMIDE

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
B0004672molecular_functionprotein kinase activity
B0005524molecular_functionATP binding
B0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue LB7 A 901
ChainResidue
ALEU595
AVAL690
AGLU691
AHIS692
AGLY693
AARG738
AASN739
ALEU741
ASER758
AGLN597
AGLY598
AVAL603
AVAL640
ALYS642
ATHR687
AGLU688
ATYR689

site_idAC2
Number of Residues17
Detailsbinding site for residue LB7 B 901
ChainResidue
BLEU595
BGLN597
BGLY598
BVAL603
BVAL640
BLYS642
BALA671
BTHR687
BGLU688
BTYR689
BVAL690
BGLU691
BGLY693
BARG738
BLEU741
BSER758
BHOH1008

site_idAC3
Number of Residues1
Detailsbinding site for residue CL B 902
ChainResidue
BLEU745

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphotyrosine => ECO:0000250|UniProtKB:Q9R117
ChainResidueDetails
ATYR604
BTYR604

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PDB entries from 2024-07-10

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