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6NVT

Crystal structure of TLA-1 extended spectrum Beta-lactamase

Functional Information from GO Data
ChainGOidnamespacecontents
A0008800molecular_functionbeta-lactamase activity
A0016787molecular_functionhydrolase activity
A0017001biological_processantibiotic catabolic process
A0030655biological_processbeta-lactam antibiotic catabolic process
A0046677biological_processresponse to antibiotic
B0008800molecular_functionbeta-lactamase activity
B0016787molecular_functionhydrolase activity
B0017001biological_processantibiotic catabolic process
B0030655biological_processbeta-lactam antibiotic catabolic process
B0046677biological_processresponse to antibiotic
C0008800molecular_functionbeta-lactamase activity
C0016787molecular_functionhydrolase activity
C0017001biological_processantibiotic catabolic process
C0030655biological_processbeta-lactam antibiotic catabolic process
C0046677biological_processresponse to antibiotic
D0008800molecular_functionbeta-lactamase activity
D0016787molecular_functionhydrolase activity
D0017001biological_processantibiotic catabolic process
D0030655biological_processbeta-lactam antibiotic catabolic process
D0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue SO4 A 301
ChainResidue
ASER70
ASER130
ATHR235
AGLY236
ASER237
AHOH409
AHOH416
AHOH458

site_idAC2
Number of Residues4
Detailsbinding site for residue SO4 A 302
ChainResidue
ATRP105
AASN132
AHIS170
ATHR104

site_idAC3
Number of Residues5
Detailsbinding site for residue SO4 A 303
ChainResidue
ALYS124
AARG129
AHOH437
AHOH522
AHOH557

site_idAC4
Number of Residues3
Detailsbinding site for residue SO4 A 304
ChainResidue
ALYS93
AHOH406
AHOH508

site_idAC5
Number of Residues6
Detailsbinding site for residue SO4 A 305
ChainResidue
ALYS98
ALYS99
ASER100
AHOH412
AHOH426
AHOH470

site_idAC6
Number of Residues2
Detailsbinding site for residue SO4 A 306
ChainResidue
AARG129
ATHR215

site_idAC7
Number of Residues3
Detailsbinding site for residue SO4 A 307
ChainResidue
APRO226
AASP227
AHOH405

site_idAC8
Number of Residues4
Detailsbinding site for residue CL A 308
ChainResidue
APHE193
AASN196
AILE198
ALEU199

site_idAC9
Number of Residues5
Detailsbinding site for residue ACT A 309
ChainResidue
AASN61
AGLU62
ALYS63
AHIS64
AACT317

site_idAD1
Number of Residues5
Detailsbinding site for residue ACT A 310
ChainResidue
AHOH417
AHOH463
AHOH521
AHOH630
DSER100

site_idAD2
Number of Residues1
Detailsbinding site for residue ACT A 311
ChainResidue
ALYS201

site_idAD3
Number of Residues5
Detailsbinding site for residue ACT A 312
ChainResidue
ALYS270
ASER271
AHOH401
DLYS93
DHOH522

site_idAD4
Number of Residues5
Detailsbinding site for residue ACT A 313
ChainResidue
ASER118
ASER120
AGLU121
AHOH415
AHOH633

site_idAD5
Number of Residues4
Detailsbinding site for residue ACT A 314
ChainResidue
AGLY217
AHOH558
AHOH559
AHOH609

site_idAD6
Number of Residues2
Detailsbinding site for residue ACT A 315
ChainResidue
ALYS195
AHOH534

site_idAD7
Number of Residues3
Detailsbinding site for residue ACT A 316
ChainResidue
ASER90
AILE91
AASN202

site_idAD8
Number of Residues5
Detailsbinding site for residue ACT A 317
ChainResidue
ALYS30
AGLU34
AASN61
AGLU62
AACT309

site_idAD9
Number of Residues6
Detailsbinding site for residue ACT A 318
ChainResidue
AGLY144
ATHR145
ATHR165
AHOH402
AHOH419
AHOH591

site_idAE1
Number of Residues4
Detailsbinding site for residue ACT A 319
ChainResidue
ALYS270
AASP272
AHOH519
DASN88

site_idAE2
Number of Residues3
Detailsbinding site for residue ACT A 320
ChainResidue
ATRP180
AHOH404
AHOH617

site_idAE3
Number of Residues4
Detailsbinding site for residue SO4 B 301
ChainResidue
BARG129
BHOH415
BHOH448
BHOH550

site_idAE4
Number of Residues3
Detailsbinding site for residue SO4 B 302
ChainResidue
BPRO226
BASP227
BHOH412

site_idAE5
Number of Residues3
Detailsbinding site for residue SO4 B 303
ChainResidue
BLYS201
BHOH446
BHOH530

site_idAE6
Number of Residues3
Detailsbinding site for residue SO4 B 304
ChainResidue
BSER90
BILE91
BHOH445

site_idAE7
Number of Residues5
Detailsbinding site for residue SO4 B 305
ChainResidue
BHIS170
BHOH425
BTHR104
BTRP105
BASN132

site_idAE8
Number of Residues7
Detailsbinding site for residue SO4 B 306
ChainResidue
BSER70
BSER130
BTHR235
BGLY236
BSER237
BHOH403
BHOH557

site_idAE9
Number of Residues4
Detailsbinding site for residue SO4 B 307
ChainResidue
BARG129
BTHR215
BHOH421
BHOH512

site_idAF1
Number of Residues4
Detailsbinding site for residue CL B 308
ChainResidue
BPHE193
BASN196
BILE198
BLEU199

site_idAF2
Number of Residues2
Detailsbinding site for residue ACT B 309
ChainResidue
BLYS98
BHOH411

site_idAF3
Number of Residues4
Detailsbinding site for residue ACT B 310
ChainResidue
BLYS30
BGLU34
BASN61
BHOH431

site_idAF4
Number of Residues4
Detailsbinding site for residue ACT B 311
ChainResidue
BLYS270
BASP272
BHOH401
BHOH438

site_idAF5
Number of Residues3
Detailsbinding site for residue ACT B 312
ChainResidue
BLYS93
BLYS94
BHOH408

site_idAF6
Number of Residues3
Detailsbinding site for residue ACT B 313
ChainResidue
BGLY217
BHOH407
BHOH646

site_idAF7
Number of Residues2
Detailsbinding site for residue ACT B 314
ChainResidue
BASP92
BSER118

site_idAF8
Number of Residues7
Detailsbinding site for residue SO4 C 301
ChainResidue
CSER70
CSER130
CTHR235
CGLY236
CSER237
CHOH407
CHOH565

site_idAF9
Number of Residues5
Detailsbinding site for residue SO4 C 302
ChainResidue
CTHR104
CTRP105
CASN132
CHIS170
CHOH555

site_idAG1
Number of Residues1
Detailsbinding site for residue SO4 C 303
ChainResidue
CHOH479

site_idAG2
Number of Residues2
Detailsbinding site for residue SO4 C 304
ChainResidue
CARG129
CHOH428

site_idAG3
Number of Residues3
Detailsbinding site for residue SO4 C 305
ChainResidue
CASP227
CHOH411
CHOH419

site_idAG4
Number of Residues6
Detailsbinding site for residue SO4 C 306
ChainResidue
CSER200
CLYS201
CHOH418
CHOH426
CHOH478
CHOH504

site_idAG5
Number of Residues2
Detailsbinding site for residue SO4 C 307
ChainResidue
CSER90
CILE91

site_idAG6
Number of Residues6
Detailsbinding site for residue SO4 C 308
ChainResidue
CLYS99
CSER100
CHOH406
CHOH455
CHOH496
CHOH503

site_idAG7
Number of Residues3
Detailsbinding site for residue SO4 C 309
ChainResidue
CARG129
CTHR215
CHOH430

site_idAG8
Number of Residues3
Detailsbinding site for residue SO4 C 310
ChainResidue
CLYS270
CSER271
CHOH402

site_idAG9
Number of Residues5
Detailsbinding site for residue CL C 311
ChainResidue
CTHR214
CTHR216
CLYS222
CHIS233
CHOH470

site_idAH1
Number of Residues5
Detailsbinding site for residue CL C 312
ChainResidue
CPRO67
CALA243
CASN245
CTYR263
CSER265

site_idAH2
Number of Residues4
Detailsbinding site for residue CL C 313
ChainResidue
CPHE193
CASN196
CILE198
CLEU199

site_idAH3
Number of Residues4
Detailsbinding site for residue CL C 314
ChainResidue
CGLY144
CTHR145
CHOH524
CHOH633

site_idAH4
Number of Residues4
Detailsbinding site for residue ACT C 315
ChainResidue
CASN114
CHOH403
CHOH511
DLYS171

site_idAH5
Number of Residues4
Detailsbinding site for residue ACT C 316
ChainResidue
CLYS93
CLYS94
CHOH487
DHOH410

site_idAH6
Number of Residues5
Detailsbinding site for residue ACT C 317
ChainResidue
CLYS30
CGLU34
CASN61
CGLU62
CHOH499

site_idAH7
Number of Residues2
Detailsbinding site for residue ACT C 318
ChainResidue
CGLY217
CHOH401

site_idAH8
Number of Residues4
Detailsbinding site for residue ACT C 319
ChainResidue
CLYS219
CLYS276
CACT320
CHOH431

site_idAH9
Number of Residues2
Detailsbinding site for residue ACT C 320
ChainResidue
CLYS276
CACT319

site_idAI1
Number of Residues2
Detailsbinding site for residue ACT C 321
ChainResidue
CASP227
CGLY228

site_idAI2
Number of Residues7
Detailsbinding site for residue SO4 D 301
ChainResidue
DSER70
DSER130
DTHR235
DGLY236
DSER237
DHOH408
DHOH567

site_idAI3
Number of Residues6
Detailsbinding site for residue SO4 D 302
ChainResidue
DTHR104
DTRP105
DASN132
DHIS170
DHOH448
DHOH483

site_idAI4
Number of Residues4
Detailsbinding site for residue SO4 D 303
ChainResidue
DLYS124
DARG129
DHOH445
DHOH465

site_idAI5
Number of Residues3
Detailsbinding site for residue SO4 D 304
ChainResidue
DPRO226
DASP227
DHOH407

site_idAI6
Number of Residues2
Detailsbinding site for residue SO4 D 305
ChainResidue
DLYS201
DHOH428

site_idAI7
Number of Residues3
Detailsbinding site for residue SO4 D 306
ChainResidue
DARG129
DTHR215
DHOH421

site_idAI8
Number of Residues2
Detailsbinding site for residue CL D 307
ChainResidue
DTHR145
DHOH498

site_idAI9
Number of Residues5
Detailsbinding site for residue CL D 308
ChainResidue
DPHE193
DASN196
DGLU197
DILE198
DLEU199

site_idAJ1
Number of Residues4
Detailsbinding site for residue ACT D 309
ChainResidue
DASP92
DSER118
DHOH402
DHOH403

site_idAJ2
Number of Residues3
Detailsbinding site for residue ACT D 310
ChainResidue
AHOH401
DLYS93
DLYS94

site_idAJ3
Number of Residues3
Detailsbinding site for residue ACT D 311
ChainResidue
DSER153
DLYS158
DASN159

site_idAJ4
Number of Residues4
Detailsbinding site for residue ACT D 312
ChainResidue
CHOH471
CHOH505
DHOH444
DHOH575

site_idAJ5
Number of Residues4
Detailsbinding site for residue ACT D 313
ChainResidue
DGLY217
DHOH412
DHOH435
DHOH640

site_idAJ6
Number of Residues6
Detailsbinding site for residue ACT D 314
ChainResidue
DLYS30
DGLU34
DASN59
DASN61
DGLU62
DHOH415

site_idAJ7
Number of Residues4
Detailsbinding site for residue ACT D 315
ChainResidue
CLYS93
DLYS270
DSER271
DHOH410

site_idAJ8
Number of Residues4
Detailsbinding site for residue ACT D 316
ChainResidue
CASN88
DLYS270
DASP272
DHOH462

site_idAJ9
Number of Residues2
Detailsbinding site for residue ACT D 317
ChainResidue
DASP227
DGLY228

site_idAK1
Number of Residues3
Detailsbinding site for residue ACT D 318
ChainResidue
DGLY25
DTHR26
DTYR288

site_idAK2
Number of Residues2
Detailsbinding site for residue ACT D 319
ChainResidue
DLYS195
DHOH598

site_idAK3
Number of Residues3
Detailsbinding site for residue ACT D 320
ChainResidue
AHIS170
ALYS171
DASN114

Functional Information from PROSITE/UniProt
site_idPS00146
Number of Residues16
DetailsBETA_LACTAMASE_A Beta-lactamase class-A active site. YpMQSTyKfhlALAVL
ChainResidueDetails
ATYR66-LEU81

221051

PDB entries from 2024-06-12

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