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6M9H

JAK2 JH2 in complex with diaminopyrimidine JAK040

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue J9D A 901
ChainResidue
ALEU579
AASN678
ALEU680
AHOH1188
AGLN626
AGLU627
APHE628
AVAL629
ALYS630
AGLY632
ASER633
ALYS677

site_idAC2
Number of Residues7
Detailsbinding site for residue GOL A 902
ChainResidue
AASN673
ACYS675
AARG715
ATRP718
AHOH1071
AHOH1091
AHOH1118

site_idAC3
Number of Residues1
Detailsbinding site for residue DMS A 903
ChainResidue
AASN667

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSite: {"description":"Breakpoint for translocation to form PCM1-JAK2 fusion protein"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsModified residue: {"description":"Phosphotyrosine","evidences":[{"source":"PubMed","id":"23186163","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

247947

PDB entries from 2026-01-21

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