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6M9H

JAK2 JH2 in complex with diaminopyrimidine JAK040

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue J9D A 901
ChainResidue
ALEU579
AASN678
ALEU680
AHOH1188
AGLN626
AGLU627
APHE628
AVAL629
ALYS630
AGLY632
ASER633
ALYS677

site_idAC2
Number of Residues7
Detailsbinding site for residue GOL A 902
ChainResidue
AASN673
ACYS675
AARG715
ATRP718
AHOH1071
AHOH1091
AHOH1118

site_idAC3
Number of Residues1
Detailsbinding site for residue DMS A 903
ChainResidue
AASN667

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Breakpoint for translocation to form PCM1-JAK2 fusion protein
ChainResidueDetails
AASP710

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphotyrosine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ATYR570

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PDB entries from 2024-07-17

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