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6LU5

Crystal structure of BPTF-BRD with ligand DCBPin5 bound

Functional Information from GO Data
ChainGOidnamespacecontents
A0006357biological_processregulation of transcription by RNA polymerase II
A0016589cellular_componentNURF complex
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue EUO A 201
ChainResidue
ATRP91
AASN148
APHE154
AHOH318
APRO92
APHE93
APRO96
AVAL97
AASP98
AASP101
ACYS144
ATYR147

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFlepvDpndap..DYYgvIkepMdlatMeervqrry..Yekltefvadmtk.IfdNCryY
ChainResidueDetails
AALA90-TYR147

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI2
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

244349

PDB entries from 2025-11-05

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