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6LOC

Crystal structure of RORgammat with ligand C46D bound

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0003824molecular_functioncatalytic activity
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues20
Detailsbinding site for residue EKL A 601
ChainResidue
ACYS285
AMET365
AARG367
AALA368
APHE377
APHE378
APHE388
AILE397
AILE400
APHE401
ATYR502
AGLN286
AHOH720
ALEU287
ALEU292
ATRP317
ACYS320
AHIS323
ALEU324
AARG364

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsMotif: {"description":"AF-2"}
ChainResidueDetails

246905

PDB entries from 2025-12-31

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