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6KKB

A novel agonist of THRb

Functional Information from GO Data
ChainGOidnamespacecontents
X0003677molecular_functionDNA binding
X0004879molecular_functionnuclear receptor activity
X0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue 8HO X 501
ChainResidue
XILE275
XLEU346
XHOH659
XHOH674
XHOH723
XILE276
XARG282
XMET313
XSER314
XALA317
XLEU330
XASN331
XGLY344

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"15466465","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1Y0X","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 3"}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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