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6KEF

BRD4 Bromodomain1 with an inhibitor

Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue D7X A 201
ChainResidue
ATRP81
AASN140
AHOH335
APRO82
AGLN85
APRO86
AVAL87
AASP88
ALEU92
AASP96
ALYS99

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

219140

PDB entries from 2024-05-01

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