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6J3O

Crystal structure of the human PCAF bromodomain in complex with compound 12

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
B0004402molecular_functionhistone acetyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue B4L A 900
ChainResidue
APRO747
APRO751
AGLU756
AASN803
ATYR809
AHOH1018

site_idAC2
Number of Residues6
Detailsbinding site for residue B4L B 900
ChainResidue
BALA757
BASN803
BTYR809
BPRO747
BPRO751
BGLU756

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFmepvKrteap..GYYevIrfpMdlktMserlknry..Yvskklfmadlqr.VftNCkeY
ChainResidueDetails
AALA745-TYR802

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PDB entries from 2024-07-17

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