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6IN2

Crystal structure of BRD1 in complex with 18-Crown-6

Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue ACT A 701
ChainResidue
AVAL591
AASN642
APHE648
AHOH807
AHOH812

site_idAC2
Number of Residues6
Detailsbinding site for residue O4B A 702
ChainResidue
AVAL662
AHIS688
AGLN577
AASP580
ALYS581
AGLN658

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AriFaqpvSlkevp..DYLdhIkhpMdfatMrkrleaqg..Yknlhefeedfdl.IidNCmkY
ChainResidueDetails
AALA584-TYR641

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS594

222624

PDB entries from 2024-07-17

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