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6I7X

Crystal Structure of the first bromodomain of BRD4 in complex with RT53

Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue EDO A 201
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 202
ChainResidue
AGLY143
AVAL147
AGLU151
AHOH305

site_idAC3
Number of Residues3
Detailsbinding site for residue EDO A 203
ChainResidue
APRO56
ALYS57
ALYS102

site_idAC4
Number of Residues14
Detailsbinding site for residue H7B A 204
ChainResidue
APRO53
ATRP81
APRO82
ALEU92
ALEU94
AASP96
ATYR139
AASN140
AASP145
AILE146
AMET149
AHOH315
AHOH345
AHOH359

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

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PDB entries from 2024-07-17

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