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6HO1

TRANSCRIPTIONAL REPRESSOR ETHR FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH BDM41974

Functional Information from GO Data
ChainGOidnamespacecontents
A0000976molecular_functiontranscription cis-regulatory region binding
A0003677molecular_functionDNA binding
A0003700molecular_functionDNA-binding transcription factor activity
A0005515molecular_functionprotein binding
A0005829cellular_componentcytosol
A0006355biological_processregulation of DNA-templated transcription
A0045892biological_processnegative regulation of DNA-templated transcription
A0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue GOL A 301
ChainResidue
APRO41
ALEU42
ALEU72
AARG122
AALA123
AALA126

site_idAC2
Number of Residues14
Detailsbinding site for residue GFW A 302
ChainResidue
AGLY106
APHE110
APHE114
ATRP145
ATYR148
ATHR149
AVAL152
AASN176
AASN179
ALEU183
ATRP207
ALEU90
AMET102
ATRP103

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues19
DetailsDNA_BIND: H-T-H motif => ECO:0000255|PROSITE-ProRule:PRU00335
ChainResidueDetails
ASER46-PHE65

site_idSWS_FT_FI2
Number of Residues2
DetailsSITE: Inhibitor-binding
ChainResidueDetails
AASN176
AASN179

222624

PDB entries from 2024-07-17

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