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6HI5

The ATAD2 bromodomain in complex with compound 8

Functional Information from GO Data
ChainGOidnamespacecontents
A0006325biological_processchromatin organization
A0006355biological_processregulation of transcription, DNA-templated
A0016887molecular_functionATP hydrolysis activity
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue SO4 A 1201
ChainResidue
AARG987
AARG990
AARG994
AARG1067
AHOH1361

site_idAC2
Number of Residues3
Detailsbinding site for residue SO4 A 1202
ChainResidue
AARG1077
AHOH1326
AHOH1341

site_idAC3
Number of Residues8
Detailsbinding site for residue G6E A 1203
ChainResidue
AALA1001
AILE1002
AARG1007
ASER1032
AILE1035
AHOH1315
AHOH1332
AHIS998

site_idAC4
Number of Residues6
Detailsbinding site for residue G6E A 1204
ChainResidue
AVAL1008
AVAL1013
AASN1064
AGLY1070
AASP1071
AHOH1313

site_idAC5
Number of Residues8
Detailsbinding site for residue G6E A 1205
ChainResidue
ASER979
AGLN981
AARG1072
AARG1075
AHIS1076
ACYS1079
AALA1080
AHOH1320

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PDB entries from 2024-07-10

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