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6H0Z

Crystal Structure of KDM4D with tetrazolylhydrazide ligand NR067

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 401
ChainResidue
ACYS238
AHIS244
ACYS310
ACYS312

site_idAC2
Number of Residues2
Detailsbinding site for residue CL A 402
ChainResidue
AASN128
ALYS186

site_idAC3
Number of Residues5
Detailsbinding site for residue NA A 403
ChainResidue
AHOH660
AHOH804
AASN17
AASN262
AHOH614

site_idAC4
Number of Residues5
Detailsbinding site for residue EDO A 404
ChainResidue
AARG123
ALYS124
ALYS127
AASN128
AHOH745

site_idAC5
Number of Residues8
Detailsbinding site for residue EDO A 405
ChainResidue
ALYS150
AGLN151
ATRP152
AASN153
AHIS156
AHOH707
AHOH715
AHOH819

site_idAC6
Number of Residues4
Detailsbinding site for residue EDO A 406
ChainResidue
APRO251
ATHR252
ALYS255
AARG263

site_idAC7
Number of Residues8
Detailsbinding site for residue EDO A 407
ChainResidue
ATYR179
ATYR181
AGLU194
ASER200
AILE293
AASN294
AFHQ412
AHOH732

site_idAC8
Number of Residues7
Detailsbinding site for residue SO4 A 408
ChainResidue
AARG60
ATHR62
AASN65
AHOH519
AHOH523
AHOH531
AHOH782

site_idAC9
Number of Residues11
Detailsbinding site for residue SO4 A 409
ChainResidue
AMET19
AILE20
ALYS255
AHOH502
AHOH589
AHOH604
AHOH648
AHOH696
AHOH722
AHOH816
AHOH899

site_idAD1
Number of Residues5
Detailsbinding site for residue NI A 410
ChainResidue
AHIS192
AGLU194
AHIS280
AFHQ412
AHOH729

site_idAD2
Number of Residues15
Detailsbinding site for residue FHQ A 411
ChainResidue
ATYR63
AARG102
AALA105
AASN106
AGLN111
ATHR112
AGLY207
AGLU208
AGLY286
APHE287
AHOH508
AHOH572
AHOH616
AHOH675
AHOH772

site_idAD3
Number of Residues15
Detailsbinding site for residue FHQ A 412
ChainResidue
ATYR136
APHE189
AHIS192
AGLU194
ASER200
AASN202
ALYS210
ATRP212
AHIS280
AEDO407
ANI410
AHOH691
AHOH729
AHOH755
AHOH850

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:B2RXH2
ChainResidueDetails
ATYR136
AASN202
ALYS210
ALYS245

site_idSWS_FT_FI2
Number of Residues3
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00538, ECO:0000305|PubMed:26741168
ChainResidueDetails
AHIS192
AGLU194
AHIS280

site_idSWS_FT_FI3
Number of Residues4
DetailsBINDING: BINDING => ECO:0007744|PDB:5F5A, ECO:0007744|PDB:5F5C
ChainResidueDetails
ACYS238
AHIS244
ACYS310
ACYS312

site_idSWS_FT_FI4
Number of Residues2
DetailsMOD_RES: PolyADP-ribosyl glutamic acid => ECO:0000269|PubMed:23102699
ChainResidueDetails
AGLU26
AGLU27

222415

PDB entries from 2024-07-10

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