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6GJ6

CRYSTAL STRUCTURE OF KRAS G12D (GPPCP) IN COMPLEX WITH 18

Functional Information from GO Data
ChainGOidnamespacecontents
A0003924molecular_functionGTPase activity
A0005525molecular_functionGTP binding
A0007165biological_processsignal transduction
A0016020cellular_componentmembrane
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue MG A 201
ChainResidue
ASER17
ATHR35
AGCP203
AHOH311
AHOH313

site_idAC2
Number of Residues10
Detailsbinding site for residue NO3 A 202
ChainResidue
AILE46
AASP47
ATYR157
AARG161
AHOH308
AHOH365
AILE24
AGLN25
AASN26
AVAL45

site_idAC3
Number of Residues30
Detailsbinding site for residue GCP A 203
ChainResidue
AASP12
AGLY13
AVAL14
AGLY15
ALYS16
ASER17
AALA18
APHE28
AVAL29
AASP30
AGLU31
ATYR32
APRO34
ATHR35
AGLY60
AASN116
ALYS117
AASP119
ALEU120
ASER145
AALA146
ALYS147
AMG201
AHOH307
AHOH311
AHOH313
AHOH342
AHOH347
AHOH354
AHOH376

site_idAC4
Number of Residues13
Detailsbinding site for residue EZZ A 204
ChainResidue
ALEU6
AVAL7
ATYR32
AGLU37
AARG41
AASP54
ALEU56
AGLN70
ATYR71
ATHR74
AHOH341
AHOH380
AHOH384

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000269|PubMed:22431598, ECO:0000269|PubMed:22566140
ChainResidueDetails
AGLY10
AVAL29
AALA59
AASN116

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: N-acetylmethionine; in GTPase KRas; alternate => ECO:0000269|Ref.17
ChainResidueDetails
AMET1

site_idSWS_FT_FI3
Number of Residues1
DetailsMOD_RES: N-acetylthreonine; in GTPase KRas, N-terminally processed => ECO:0000269|Ref.17
ChainResidueDetails
ATHR2

site_idSWS_FT_FI4
Number of Residues1
DetailsMOD_RES: N6-acetyllysine => ECO:0000269|PubMed:22711838
ChainResidueDetails
ALYS104

site_idSWS_FT_FI5
Number of Residues1
DetailsCARBOHYD: (Microbial infection) O-linked (Glc) threonine; by P.sordellii toxin TcsL => ECO:0000269|PubMed:19744486
ChainResidueDetails
ATHR35

223166

PDB entries from 2024-07-31

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