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6G34

Crystal structure of haspin in complex with 5-iodotubercidin

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue 5ID A 401
ChainResidue
AILE49
AGLY212
ALEU215
AILE245
AIOD402
AHOH512
AHOH535
AHOH571
AHOH640
AGLY50
AALA68
APHE164
AGLU165
APHE166
AGLY167
AGLY168
AASP170

site_idAC2
Number of Residues2
Detailsbinding site for residue IOD A 402
ChainResidue
ALYS70
A5ID401

site_idAC3
Number of Residues6
Detailsbinding site for residue EPE A 403
ChainResidue
AGLU287
AASN289
AHIS296
ALEU341
AASN342
APHE343

site_idAC4
Number of Residues5
Detailsbinding site for residue PO4 A 404
ChainResidue
AILE96
APRO130
AARG254
AILE257
AHOH656

Functional Information from PROSITE/UniProt
site_idPS00107
Number of Residues22
DetailsPROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. IGEGVFGEVFqTiadhtp............VAIK
ChainResidueDetails
AILE49-LYS70

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues314
DetailsDomain: {"description":"Protein kinase","evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"},{"evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsActive site: {"description":"Proton acceptor","evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues9
DetailsBinding site: {"evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues10
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"19918057","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"3DLZ","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"19918057","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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