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6G0G

BRD4 (BD1) in complex with APSC-derived ligands (e.g. sulfasalazine)

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue EDO A 201
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135
AHOH334

site_idAC2
Number of Residues4
Detailsbinding site for residue FMT A 202
ChainResidue
AHOH354
AASN44
AASP88
AASN162

site_idAC3
Number of Residues5
Detailsbinding site for residue DMS A 203
ChainResidue
ALEU94
AASN140
ASAS204
ASAS204
AHOH308

site_idAC4
Number of Residues14
Detailsbinding site for residue SAS A 204
ChainResidue
ATRP81
ATRP81
APRO82
APRO82
ALEU92
AASP145
AMET149
AMET149
ADMS203
ADMS203
AHOH335
AHOH340
AHOH344
AHOH382

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues106
DetailsDomain: {"description":"Bromo 1","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsSite: {"description":"Acetylated histone binding","evidences":[{"source":"PubMed","id":"22464331","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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