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6FGL

Crystal Structure of BAZ2A bromodomain in complex with acetylindole compound UZH47

Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue UO1 A 1901
ChainResidue
ATRP1816
AHOH2035
APRO1817
AGLU1820
APRO1821
AVAL1822
AASN1823
ALEU1826
AASN1873
AHOH2024

site_idAC2
Number of Residues6
Detailsbinding site for residue MG A 1902
ChainResidue
AHOH2005
AHOH2008
AHOH2046
AHOH2062
AHOH2095
AHOH2097

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFlepvNprlvs..GYRriIknpMdfstMrerllrgg..Ytsseefaadall.VfdNCqtF
ChainResidueDetails
AALA1815-PHE1872

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PDB entries from 2024-09-11

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