6FE6
Solution structure of a last generation P2-P4 macrocyclic inhibitor
Functional Information from GO Data
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 18 |
Details | binding site for residue 4P2 A 201 |
Chain | Residue |
A | GLN41 |
A | GLY137 |
A | SER139 |
A | PHE154 |
A | ARG155 |
A | ALA156 |
A | ALA157 |
A | VAL158 |
A | CYS159 |
A | ASP168 |
A | SER42 |
A | TYR56 |
A | HIS57 |
A | VAL78 |
A | ASP81 |
A | VAL132 |
A | LEU135 |
A | LYS136 |
site_id | AC2 |
Number of Residues | 5 |
Details | binding site for residue ZN A 202 |
Chain | Residue |
A | CYS97 |
A | CYS99 |
A | CYS145 |
A | SER147 |
A | HIS149 |