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6F5T

Crystal Structure of KDM4D with tetrazole ligand GF057

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 401
ChainResidue
ACYS238
AHIS244
ACYS310
ACYS312

site_idAC2
Number of Residues5
Detailsbinding site for residue SO4 A 402
ChainResidue
AARG102
AHIS103
AASN106
AHOH501
AHOH507

site_idAC3
Number of Residues5
Detailsbinding site for residue SO4 A 403
ChainResidue
AASN65
AILE66
ASER67
AARG102
AHOH643

site_idAC4
Number of Residues6
Detailsbinding site for residue SO4 A 404
ChainResidue
APRO113
ALYS124
AASN128
ATRP185
ALYS186
AHOH608

site_idAC5
Number of Residues4
Detailsbinding site for residue SO4 A 405
ChainResidue
AARG123
ALYS124
ALYS127
AASN128

site_idAC6
Number of Residues5
Detailsbinding site for residue NI A 406
ChainResidue
AHIS192
AGLU194
AHIS280
ACQK407
AHOH544

site_idAC7
Number of Residues15
Detailsbinding site for residue CQK A 407
ChainResidue
ATYR136
ATYR181
APHE189
AHIS192
AGLU194
ALYS210
ATRP212
ALYS245
AHIS280
ANI406
AHOH518
AHOH544
AHOH605
AHOH652
AHOH720

site_idAC8
Number of Residues14
Detailsbinding site for residue EPE A 408
ChainResidue
APHE21
AHIS22
ATYR34
ATYR37
AGLN41
AGLU256
AGLY258
AEPE409
AHOH513
AHOH586
AHOH612
AHOH666
AHOH787
AHOH795

site_idAC9
Number of Residues6
Detailsbinding site for residue EPE A 409
ChainResidue
AGLU27
ALYS33
ATYR34
ATYR37
AEPE408
AHOH589

site_idAD1
Number of Residues3
Detailsbinding site for residue EDO A 410
ChainResidue
AMET306
AHOH531
AHOH786

site_idAD2
Number of Residues3
Detailsbinding site for residue EDO A 411
ChainResidue
AARG263
AILE264
ATHR265

site_idAD3
Number of Residues6
Detailsbinding site for residue EDO A 412
ChainResidue
APHE28
AASP30
APHE31
AGLN151
ATRP152
AHOH746

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:B2RXH2
ChainResidueDetails
ALYS245
ATYR136
AASN202
ALYS210

site_idSWS_FT_FI2
Number of Residues3
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00538, ECO:0000305|PubMed:26741168
ChainResidueDetails
AHIS192
AGLU194
AHIS280

site_idSWS_FT_FI3
Number of Residues4
DetailsBINDING: BINDING => ECO:0007744|PDB:5F5A, ECO:0007744|PDB:5F5C
ChainResidueDetails
AHIS244
ACYS310
ACYS312
ACYS238

site_idSWS_FT_FI4
Number of Residues2
DetailsMOD_RES: PolyADP-ribosyl glutamic acid => ECO:0000269|PubMed:23102699
ChainResidueDetails
AGLU26
AGLU27

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PDB entries from 2024-06-12

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