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6EWF

Leishmania major N-myristoyltransferase with bound myristoyl-CoA and inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004379molecular_functionglycylpeptide N-tetradecanoyltransferase activity
A0005737cellular_componentcytoplasm
A0006499biological_processN-terminal protein myristoylation
A0016746molecular_functionacyltransferase activity
A0046872molecular_functionmetal ion binding
Functional Information from PDB Data
site_idAC1
Number of Residues32
Detailsbinding site for residue MYA A 501
ChainResidue
AHIS12
ACYS170
AVAL171
AARG176
AGLU177
ALYS178
AARG179
ALEU180
AALA181
APRO182
ATHR189
AALA13
AVAL192
ATRP198
AALA200
ATYR202
ATHR203
ALEU208
ATYR404
AHOH604
AHOH620
AHOH625
APHE14
AHOH680
AHOH682
AHOH691
ATRP15
AASN79
ATYR80
AVAL81
APHE168
ALEU169

site_idAC2
Number of Residues13
Detailsbinding site for residue 31A A 502
ChainResidue
AVAL81
AASP83
APHE88
APHE90
ATYR92
ATYR217
ATYR326
ASER330
ALEU341
ATYR345
AMET377
AMET420
ALEU421

Functional Information from PROSITE/UniProt
site_idPS00975
Number of Residues9
DetailsNMT_1 Myristoyl-CoA:protein N-myristoyltransferase signature 1. EINFLCvHK
ChainResidueDetails
AGLU165-LYS173

site_idPS00976
Number of Residues7
DetailsNMT_2 Myristoyl-CoA:protein N-myristoyltransferase signature 2. KFGaGDG
ChainResidueDetails
ALYS391-GLY397

224004

PDB entries from 2024-08-21

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