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6EPX

The ATAD2 bromodomain in complex with compound 3

Functional Information from GO Data
ChainGOidnamespacecontents
A0006325biological_processchromatin organization
A0006355biological_processregulation of transcription, DNA-templated
A0016887molecular_functionATP hydrolysis activity
Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue BQW A 1201
ChainResidue
AVAL1013
ATYR1063
AASN1064
AGLY1070
AASP1071
AHOH1304
AHOH1340

site_idAC2
Number of Residues5
Detailsbinding site for residue BQW A 1202
ChainResidue
AASP1083
AHOH1303
AHOH1331
AGLU982
ACYS1079

site_idAC3
Number of Residues4
Detailsbinding site for residue SO4 A 1203
ChainResidue
AARG987
AARG990
AARG994
AARG1067

218853

PDB entries from 2024-04-24

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