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6DUP

CRYSTAL STRUCTURE OF PXR IN COMPLEX WITH COMPOUND 7

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue HCJ A 501
ChainResidue
AMET243
AHIS407
ALEU411
AMET425
APHE429
AMET246
ASER247
APHE251
APHE281
AGLN285
APHE288
ATRP299
AMET323

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
BSER262
BPRO384
AASN224
ASER262
APRO384
BASN224

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PDB entries from 2024-06-12

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