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6DIS

Crystal structure of HCV NS3/4A protease in complex with P4-1 (AJ-71)

Functional Information from GO Data
ChainGOidnamespacecontents
A0006508biological_processproteolysis
A0008233molecular_functionpeptidase activity
A0008236molecular_functionserine-type peptidase activity
A0016020cellular_componentmembrane
A0019062biological_processvirion attachment to host cell
A0019087biological_processtransformation of host cell by virus
A0033644cellular_componenthost cell membrane
A0044423cellular_componentvirion component
A0046718biological_processsymbiont entry into host cell
A0046872molecular_functionmetal ion binding
Functional Information from PDB Data
site_idAC1
Number of Residues27
Detailsbinding site for residue GKG A 1201
ChainResidue
AHIS982
ALYS1136
AGLY1137
ASER1138
ASER1139
APHE1154
AARG1155
AALA1156
AALA1157
AVAL1158
AASP1168
AGLN1041
ASO41202
AHOH1373
AHOH1374
AHOH1403
AHOH1427
AHOH1441
AHOH1445
AHOH1467
APHE1043
ATYR1056
AHIS1057
AVAL1078
AASP1081
AARG1123
ALEU1135

site_idAC2
Number of Residues9
Detailsbinding site for residue SO4 A 1202
ChainResidue
ATYR1006
AGLN1008
ATYR1056
AGKG1201
AHOH1330
AHOH1357
AHOH1366
AHOH1384
AHOH1418

site_idAC3
Number of Residues7
Detailsbinding site for residue SO4 A 1203
ChainResidue
AARG1109
AHIS1110
AHOH1312
AHOH1317
AHOH1349
AHOH1394
AHOH1426

site_idAC4
Number of Residues5
Detailsbinding site for residue SO4 A 1204
ChainResidue
ALYS1080
AARG1155
APRO1171
ASER1174
AHOH1415

site_idAC5
Number of Residues7
Detailsbinding site for residue SO4 A 1205
ChainResidue
ATHR1040
AGLN1041
AARG1062
AHOH1303
AHOH1310
AHOH1332
AHOH1428

site_idAC6
Number of Residues4
Detailsbinding site for residue ZN A 1206
ChainResidue
ACYS1097
ACYS1099
ACYS1145
AHIS1149

site_idAC7
Number of Residues5
Detailsbinding site for residue GOL A 1207
ChainResidue
ALYS989
AGLY990
ASER1020
AALA1039
AARG1062

221051

PDB entries from 2024-06-12

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