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6DFN

Crystal structure of estrogen receptor alpha in complex with receptor degrader 16aa

Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue G9J A 601
ChainResidue
ALEU346
AHOH714
ATHR347
AALA350
AGLU353
ALEU387
AARG394
AMET421
AILE424
AVAL533

site_idAC2
Number of Residues3
Detailsbinding site for residue NI A 602
ChainResidue
AHIS501
BLEU497
BHIS501

site_idAC3
Number of Residues16
Detailsbinding site for residue G91 B 601
ChainResidue
BLEU346
BTHR347
BLEU349
BALA350
BASP351
BGLU353
BTRP383
BLEU384
BMET388
BARG394
BMET421
BILE424
BGLY521
BHIS524
BLEU525
BG9J602

site_idAC4
Number of Residues11
Detailsbinding site for residue G9J B 602
ChainResidue
BLEU346
BTHR347
BALA350
BGLU353
BLEU387
BARG394
BPHE404
BMET421
BILE424
BG91601
BHOH705

site_idAC5
Number of Residues5
Detailsbinding site for residue GOL B 603
ChainResidue
AHOH708
BALA322
BPRO325
BHIS356
BARG363

site_idAC6
Number of Residues8
Detailsbinding site for residue GOL B 604
ChainResidue
ASER512
BGLU385
BILE452
BASN455
BSER456
BLEU511
BILE514
BARG515

site_idAC7
Number of Residues11
Detailsbinding site for residue G9J C 601
ChainResidue
CLEU346
CTHR347
CALA350
CGLU353
CLEU387
CARG394
CPHE404
CMET421
CGLY521
CHIS524
CVAL533

site_idAC8
Number of Residues10
Detailsbinding site for residue G9J D 601
ChainResidue
DLEU346
DTHR347
DGLU353
DLEU387
DARG394
DMET421
DGLY521
DHIS524
DG91602
DHOH707

site_idAC9
Number of Residues14
Detailsbinding site for residue G91 D 602
ChainResidue
DLEU346
DTHR347
DLEU349
DALA350
DASP351
DGLU353
DLEU391
DARG394
DILE424
DLEU428
DHIS524
DLEU525
DVAL534
DG9J601

site_idAD1
Number of Residues3
Detailsbinding site for residue GOL D 603
ChainResidue
DALA322
DHIS356
DARG363

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsMOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106
ChainResidueDetails
ATYR537
BTYR537
CTYR537
DTYR537

site_idSWS_FT_FI2
Number of Residues4
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
ACYS447
BCYS447
CCYS447
DCYS447

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PDB entries from 2024-07-17

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