Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

6DDJ

Crystal Structure of the human BRD2 BD2 bromodimain in complex with a Tetrahydroquinoline analogue

Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue G7V A 501
ChainResidue
ATRP370
AHOH706
APRO371
ALEU383
AASN429
AHIS433
AVAL435
AHOH608
AHOH676
AHOH688

site_idAC2
Number of Residues7
Detailsbinding site for residue EDO A 502
ChainResidue
ATYR368
ALYS402
AASP407
AGLU413
AMET438
ALYS441
AHOH614

site_idAC3
Number of Residues7
Detailsbinding site for residue EDO A 503
ChainResidue
ATYR426
AARG440
AGLN443
AGLN443
AASP444
APHE448
AHOH636

site_idAC4
Number of Residues3
Detailsbinding site for residue EDO A 504
ChainResidue
ALEU350
AHOH603
AHOH669

site_idAC5
Number of Residues7
Detailsbinding site for residue EDO A 505
ChainResidue
AILE389
AILE390
ALYS391
AHIS392
AASN424
ALYS427
AASP455

site_idAC6
Number of Residues5
Detailsbinding site for residue EDO A 506
ChainResidue
ALEU361
ATYR373
AHOH666
AHOH690
AHOH699

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

222624

PDB entries from 2024-07-17

PDB statisticsPDBj update infoContact PDBjnumon