Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

6DDI

Crystal Structure of the human BRD2 BD1 bromodomain in complex with a Tetrahydroquinoline analogue

Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue G7V A 301
ChainResidue
ATRP97
AHOH456
AHOH466
AHOH480
BGLN94
APRO98
APHE99
ALYS107
ALEU108
ALEU110
ACYS152
AASN156
AHOH412

site_idAC2
Number of Residues3
Detailsbinding site for residue SO4 A 302
ChainResidue
AARG100
AHOH408
AHOH446

site_idAC3
Number of Residues4
Detailsbinding site for residue EDO A 303
ChainResidue
AASP160
AASP161
AILE162
AHOH464

site_idAC4
Number of Residues5
Detailsbinding site for residue EDO A 304
ChainResidue
AGLN94
ATRP97
BGLN94
BTRP97
BMET165

site_idAC5
Number of Residues11
Detailsbinding site for residue G7V B 301
ChainResidue
AGLN94
BTRP97
BPRO98
BPHE99
BLEU110
BCYS152
BASN156
BHOH413
BHOH445
BHOH448
BHOH460

site_idAC6
Number of Residues7
Detailsbinding site for residue 03S B 302
ChainResidue
BTRP97
BARG100
BHOH407
BHOH424
BHOH462
CASN132
CTYR134

site_idAC7
Number of Residues5
Detailsbinding site for residue EDO B 303
ChainResidue
BASP160
BASP161
BILE162
BHOH403
BHOH409

site_idAC8
Number of Residues10
Detailsbinding site for residue G7V C 301
ChainResidue
AGLN80
ALYS84
APRO181
CTRP97
CPRO98
CGLN101
CLEU110
CASN156
CHOH407
CHOH439

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFrqpvDavklglpDYHkiIkqpMdmgtIkrrlenny..Ywaasecmqdfnt.MftNCyiY
ChainResidueDetails
AALA96-TYR155

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:37731000, ECO:0007744|PDB:8SB6
ChainResidueDetails
ATHR159
BTHR159
CTHR159

site_idSWS_FT_FI2
Number of Residues3
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:19690332
ChainResidueDetails
ALYS84
BLYS84
CLYS84

222624

PDB entries from 2024-07-17

PDB statisticsPDBj update infoContact PDBjnumon