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6CZV

BRD4(BD1) complexed with 2759

Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue FOY A 201
ChainResidue
ATRP81
APRO82
APHE83
ALEU94
ALYS99
AASN140
AHOH311

site_idAC2
Number of Residues9
Detailsbinding site for residue EDO A 202
ChainResidue
ALEU63
AARG113
AASN117
ATYR118
ATYR119
AHOH307
AHOH309
AARG58
AGLN59

site_idAC3
Number of Residues7
Detailsbinding site for residue EDO A 203
ChainResidue
AHIS77
AGLN78
AGLU154
ALEU158
AHOH306
AHOH320
AHOH410

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

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PDB entries from 2024-07-17

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