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6C1C

FGFR1 kinase complex with inhibitor SN37116

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0004672molecular_functionprotein kinase activity
A0004713molecular_functionprotein tyrosine kinase activity
A0005007molecular_functionfibroblast growth factor receptor activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
B0004672molecular_functionprotein kinase activity
B0004713molecular_functionprotein tyrosine kinase activity
B0005007molecular_functionfibroblast growth factor receptor activity
B0005524molecular_functionATP binding
B0006468biological_processprotein phosphorylation
PDBデータベースに由来する情報
site_idAC1
残基数16
詳細binding site for residue YY6 A 801
鎖名残基
ALEU484
AGLY567
AASN568
AGLU571
AALA640
AASP641
APHE642
AHOH918
AVAL492
AALA512
ALYS514
AGLU531
AVAL559
AVAL561
AGLU562
AALA564

site_idAC2
残基数11
詳細binding site for residue YY6 B 801
鎖名残基
BLEU484
BLYS514
BGLU531
BVAL559
BVAL561
BGLU562
BALA564
BGLU571
BLEU630
BALA640
BASP641

site_idAC3
残基数3
詳細binding site for residue SO4 B 802
鎖名残基
BLYS665
BPRO702
BGLY703

UniProtにおけるモチーフ・データベースPROSITEからの機能情報
site_idPS00107
残基数31
詳細PROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. LGEGAFGQVVlAeaigldkdkpnrvtk...VAVK
鎖名残基詳細
ALEU484-LYS514

site_idPS00109
残基数13
詳細PROTEIN_KINASE_TYR Tyrosine protein kinases specific active-site signature. CIHrDLAARNVLV
鎖名残基詳細
ACYS619-VAL631

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数2
詳細ACT_SITE: Proton acceptor => ECO:0000255|PROSITE-ProRule:PRU00159, ECO:0000255|PROSITE-ProRule:PRU10028, ECO:0000269|PubMed:19224897
鎖名残基詳細
AALA625
BALA625

site_idSWS_FT_FI2
残基数12
詳細BINDING:
鎖名残基詳細
AGLU486
BARG570
BVAL629
BGLY643
ALEU516
AALA564
AARG570
AVAL629
AGLY643
BGLU486
BLEU516
BALA564

site_idSWS_FT_FI3
残基数6
詳細MOD_RES: Phosphotyrosine; by autocatalysis => ECO:0000269|PubMed:16507368, ECO:0000269|PubMed:19224897, ECO:0000269|PubMed:8622701
鎖名残基詳細
ALEU465
ATYR585
APRO587
BLEU465
BTYR585
BPRO587

site_idSWS_FT_FI4
残基数4
詳細MOD_RES: Phosphotyrosine; by autocatalysis => ECO:0000269|PubMed:16507368, ECO:0000269|PubMed:19224897, ECO:0000269|PubMed:19665973, ECO:0000269|PubMed:8622701
鎖名残基詳細
ALYS655
ALYS656
BLYS655
BLYS656

site_idSWS_FT_FI5
残基数2
詳細MOD_RES: Phosphotyrosine; by autocatalysis => ECO:0000269|PubMed:19224897, ECO:0000269|PubMed:8622701
鎖名残基詳細
AMET732
BMET732

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件を2024-09-18に公開中

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