6BQA
BRD9 bromodomain in complex with 3-(6-(but-3-en-1-yl)-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)-N,N-dimethylbenzamide
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 9 |
Details | binding site for residue 67C A 201 |
Chain | Residue |
A | PHE44 |
A | PHE45 |
A | VAL49 |
A | ILE53 |
A | ASN100 |
A | TYR106 |
A | LYS111 |
A | HOH305 |
A | HOH408 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 2 |
Details | SITE: Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding => ECO:0000269|PubMed:26365797 |
Chain | Residue | Details |
A | ILE53 | |
A | TYR106 |