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6BNS

STRUCTURE OF HUMAN PREGNANE X RECEPTOR LIGAND BINDING DOMAIN BOUND TETHERED WITH SRC co-activator peptide and Compound 25a AKA BICYCLIC HEXAFLUOROISOPROPYL 2 ALCOHOL SULFONAMIDES

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue XGH A 501
ChainResidue
ALEU206
ALEU411
APHE420
AMET425
AHOH620
ALEU209
AVAL211
AILE236
ALEU239
ALEU240
AMET243
ASER247
AHIS407

site_idAC2
Number of Residues17
Detailsbinding site for residue XGH B 501
ChainResidue
BLEU206
BLEU209
BLYS210
BVAL211
BILE236
BLEU239
BLEU240
BMET243
BSER247
BPHE288
BTRP299
BTYR306
BMET323
BHIS407
BPHE420
BMET425
BHOH606

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
ASER247
AGLN285
AHIS407
BSER247
BGLN285
BHIS407

site_idSWS_FT_FI2
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ASER460
BSER460

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PDB entries from 2024-05-01

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