6AU0
Crystal structure of PPK2 (Class III) in complex with bisphosphonate inhibitor (2-((3,5-dichlorophenyl)amino)ethane-1,1-diyl)diphosphonic acid
Functional Information from GO Data
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 12 |
Details | binding site for residue BWJ A 401 |
Chain | Residue |
A | ALA78 |
A | ASP222 |
A | HOH559 |
A | HOH561 |
A | ALA79 |
A | GLY80 |
A | LYS81 |
A | ASP82 |
A | GLY83 |
A | ARG204 |
A | PHE205 |
A | ARG208 |
site_id | AC2 |
Number of Residues | 7 |
Details | binding site for residue GOL A 402 |
Chain | Residue |
A | HIS195 |
A | SER197 |
A | LYS198 |
A | TRP229 |
A | ARG233 |
A | HOH509 |
A | HOH544 |
site_id | AC3 |
Number of Residues | 7 |
Details | binding site for residue GOL A 403 |
Chain | Residue |
A | TYR114 |
A | SER155 |
A | PHE167 |
A | ARG171 |
A | GLN174 |
A | GLU184 |
A | ASN185 |