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6AJW

Crystal structure of BRD4 in complex with DMSO (Cocktail No. 4)

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue NA A 201
ChainResidue
AVAL90
AASN93
AHOH315
AHOH330
AHOH416
AHOH423

site_idAC2
Number of Residues3
Detailsbinding site for residue DMS A 202
ChainResidue
AASN140
AILE146
AHOH311

site_idAC3
Number of Residues6
Detailsbinding site for residue NA A 203
ChainResidue
ATYR65
ALYS160
AGLU163
AHOH363
AHOH390
AHOH419

site_idAC4
Number of Residues6
Detailsbinding site for residue NA A 204
ChainResidue
AARG58
ALEU63
AASN117
ATYR118
ATYR119
AHOH393

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

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PDB entries from 2024-07-24

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