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5ZQO

Tankyrase-2 in complex with compound 1a

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 1201
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues9
Detailsbinding site for residue 9GX A 1202
ChainResidue
APHE1061
AALA1062
ASER1068
ATYR1071
AHIS1031
AGLY1032
AALA1049
ATYR1050
ATYR1060

site_idAC3
Number of Residues9
Detailsbinding site for residue SO4 A 1203
ChainResidue
AARG977
AHIS979
AARG980
ALYS1067
AGLN1070
AHOH1304
AHOH1346
AHOH1382
BHOH1322

site_idAC4
Number of Residues6
Detailsbinding site for residue SO4 A 1204
ChainResidue
AASN990
AARG991
BPRO1160
BGLU1161
BHOH1303
BHOH1311

site_idAC5
Number of Residues7
Detailsbinding site for residue GOL A 1205
ChainResidue
ATYR1050
AGLY1053
AMET1054
ATYR1060
ATYR1071
AHOH1346
BGLU1138

site_idAC6
Number of Residues4
Detailsbinding site for residue GOL A 1206
ChainResidue
ACYS1001
ATRP1006
AHOH1325
BTYR1148

site_idAC7
Number of Residues7
Detailsbinding site for residue SO4 B 1201
ChainResidue
BHIS1117
BSER1118
BARG1143
BHOH1315
BHOH1316
BHOH1317
BHOH1319

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092

221051

PDB entries from 2024-06-12

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