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5Z8G

BRD4 Bromodomain 1 with an inhibitor

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue 99L A 201
ChainResidue
ATRP81
AMET149
AHOH311
AHOH322
APRO82
APHE83
AVAL87
AASP96
ATYR97
ATYR139
AASN140
AASP145

site_idAC2
Number of Residues7
Detailsbinding site for residue DMS A 202
ChainResidue
ATHR60
AGLN62
AASN121
AALA122
AGLU167
AHOH306
AHOH353

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

222415

PDB entries from 2024-07-10

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