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5Z8G

BRD4 Bromodomain 1 with an inhibitor

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue 99L A 201
ChainResidue
ATRP81
AMET149
AHOH311
AHOH322
APRO82
APHE83
AVAL87
AASP96
ATYR97
ATYR139
AASN140
AASP145

site_idAC2
Number of Residues7
Detailsbinding site for residue DMS A 202
ChainResidue
ATHR60
AGLN62
AASN121
AALA122
AGLU167
AHOH306
AHOH353

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues106
DetailsDomain: {"description":"Bromo 1","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsSite: {"description":"Acetylated histone binding","evidences":[{"source":"PubMed","id":"22464331","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

247947

PDB entries from 2026-01-21

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