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5Z6S

Crystal structure of the PPARgamma-LBD complexed with compound DS-6930

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue RTF A 501
ChainResidue
AILE249
ATYR327
AILE341
AMET348
APHE363
AMET364
ALYS367
AHOH643
AHOH677
ALEU255
AGLY258
AGLU259
AARG280
AILE281
AGLY284
ACYS285
ASER289

site_idAC2
Number of Residues3
Detailsbinding site for residue CL A 502
ChainResidue
AASN335
AASN375
AHOH718

site_idAC3
Number of Residues2
Detailsbinding site for residue CL A 503
ChainResidue
AARG397
APRO398

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: N6-acetyllysine => ECO:0000250|UniProtKB:O70343
ChainResidueDetails
CLYS11
AHIS323
AHIS449
ATYR473

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
ChainResidueDetails
ALYS224

223790

PDB entries from 2024-08-14

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