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5Z5T

The first bromodomain of BRD4 with compound BDF-2141

Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue 96R A 201
ChainResidue
ATRP81
AHOH309
AHOH369
APHE83
AVAL87
ALEU92
ATYR97
ACYS136
ATYR139
AASN140
AILE146

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

223532

PDB entries from 2024-08-07

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