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5YXL

A ligand M binding to FXR

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
A0032052molecular_functionbile acid binding
A0038183biological_processbile acid signaling pathway
C0003677molecular_functionDNA binding
C0004879molecular_functionnuclear receptor activity
C0006355biological_processregulation of DNA-templated transcription
C0032052molecular_functionbile acid binding
C0038183biological_processbile acid signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue NIW A 301
ChainResidue
APHE41
AHIS204
AMET207
AVAL213
ATRP226
ATHR45
AHIS51
AMET85
APHE86
ASER89
AILE114
ATYR118
AMET122

site_idAC2
Number of Residues15
Detailsbinding site for residue NIW C 301
ChainResidue
CPHE41
CLEU44
CTHR45
CALA48
CHIS51
CMET85
CPHE86
CILE114
CTYR118
CMET122
CPHE200
CHIS203
CHIS204
CMET207
CTRP226

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBinding site: {"evidences":[{"source":"PDB","id":"6HL1","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsModified residue: {"description":"Phosphothreonine; by PKC/PRKCZ","evidences":[{"source":"PubMed","id":"18668687","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO1)","evidences":[{"source":"PubMed","id":"23546875","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 3"}
ChainResidueDetails

249697

PDB entries from 2026-02-25

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