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5XPN

Crystal structure of VDR-LBD complexed with 25RS-(hydroxyphenyl)-25-methoxy-2-methylidene-19,26,27-trinor-1-hydroxyvitamin D3

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue 8BO A 501
ChainResidue
ATYR143
AVAL296
AALA299
AGLY300
AHIS301
AHIS393
AGLN396
ALEU400
A9RO502
ALEU223
AVAL230
ASER233
AARG270
ASER271
ASER274
ATRP282
ACYS284

site_idAC2
Number of Residues17
Detailsbinding site for residue 9RO A 502
ChainResidue
ATYR143
ALEU223
AVAL230
ASER233
AARG270
ASER271
ASER274
ATRP282
ACYS284
AVAL296
AALA299
AGLY300
AHIS301
AHIS393
AGLN396
ALEU400
A8BO501

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues18
DetailsRegion: {"description":"Interaction with coactivator LXXLL motif","evidences":[{"source":"PubMed","id":"15065852","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"15065852","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1RK3","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 2"}
ChainResidueDetails

248335

PDB entries from 2026-01-28

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