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5XPM

Crystal structure of VDR-LBD complexed with 22S-Butyl-25RS-(hydroxyphenyl)-25-methoxy-2-methylidene-19,26,27-trinor-1-hydroxyvitamin D3

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue 8C0 A 501
ChainResidue
ATYR143
AHIS301
ALEU305
ALEU389
AHIS393
ALEU400
APHE418
AVAL230
ASER233
AARG270
ASER271
ASER274
ATRP282
ACYS284
AALA299

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:15065852, ECO:0007744|PDB:1RK3
ChainResidueDetails
ATYR143
AMET280
ALYS317
ALEU321
AVAL348

222624

PDB entries from 2024-07-17

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